Drugs That Interact with Grapefruit Juice

 

androgen hormone inhibitor finasteride
anticoagulant warfarin
antiepileptic carbamazepine
anti-infectives albendazole, amprenavir, artemether, clarithromycin, erythromycin, halofantrine, indinavir, itraconazole, nelfinavir, praziquantil, ritonavir, saquinavir, troleandomycin
anti-inflammatories cortisol, methylprednisolone
antihyperlipidemics atorvastatin, fluvastatin, lovastatin, simvastatin
antineoplastics cyclophosphamide, etoposide, ifosfamide, tamoxifen, vinblastine, vincristine
antitussive dextromethorphan
cardiovascular agents amiodarone, cavedilol, diltiazem, felodipine, nifedipine, nimodipine, nicardipine, nisoldipine, nitrendipine, quinidine, verapamil
central nervous system agents alprazolam, amitriptyline, buspirone, carbamazepine, diazepam, fluvoxamine, midazolam, scopolamine, sertraline, triazolam
hormone ethinylestradiol, progesterone, testosterone
gastrointestinal agents cisapride
histamine H1 antagonists astemizole, fexofenadine, terfenadine
immunosuppressives cyclosporine, sirolimus, tacrolimus
opoid analgesics alfentanil, fentanyl, sufentanil
xanthine theophylline
erectile dysfunction drugs sildenafil, tadalafil

From “The Grapefruit Challenge,”AJN, Dec. 2004 & The Handbook of Drug-Nutrient Interaction, 2004