Drugs That Interact with Grapefruit Juice

 

androgen hormone inhibitorfinasteride
anticoagulantwarfarin
antiepilepticcarbamazepine
anti-infectivesalbendazole, amprenavir, artemether, clarithromycin, erythromycin, halofantrine, indinavir, itraconazole, nelfinavir, praziquantil, ritonavir, saquinavir, troleandomycin
anti-inflammatoriescortisol, methylprednisolone
antihyperlipidemicsatorvastatin, fluvastatin, lovastatin, simvastatin
antineoplasticscyclophosphamide, etoposide, ifosfamide, tamoxifen, vinblastine, vincristine
antitussivedextromethorphan
cardiovascular agentsamiodarone, cavedilol, diltiazem, felodipine, nifedipine, nimodipine, nicardipine, nisoldipine, nitrendipine, quinidine, verapamil
central nervous system agentsalprazolam, amitriptyline, buspirone, carbamazepine, diazepam, fluvoxamine, midazolam, scopolamine, sertraline, triazolam
hormoneethinylestradiol, progesterone, testosterone
gastrointestinal agentscisapride
histamine H1 antagonistsastemizole, fexofenadine, terfenadine
immunosuppressivescyclosporine, sirolimus, tacrolimus
opoid analgesics alfentanil, fentanyl, sufentanil
xanthinetheophylline
erectile dysfunction drugssildenafil, tadalafil

From “The Grapefruit Challenge,”AJN, Dec. 2004 & The Handbook of Drug-Nutrient Interaction, 2004