androgen hormone inhibitor | finasteride |
anticoagulant | warfarin |
antiepileptic | carbamazepine |
anti-infectives | albendazole, amprenavir, artemether, clarithromycin, erythromycin, halofantrine, indinavir, itraconazole, nelfinavir, praziquantil, ritonavir, saquinavir, troleandomycin |
anti-inflammatories | cortisol, methylprednisolone |
antihyperlipidemics | atorvastatin, fluvastatin, lovastatin, simvastatin |
antineoplastics | cyclophosphamide, etoposide, ifosfamide, tamoxifen, vinblastine, vincristine |
antitussive | dextromethorphan |
cardiovascular agents | amiodarone, cavedilol, diltiazem, felodipine, nifedipine, nimodipine, nicardipine, nisoldipine, nitrendipine, quinidine, verapamil |
central nervous system agents | alprazolam, amitriptyline, buspirone, carbamazepine, diazepam, fluvoxamine, midazolam, scopolamine, sertraline, triazolam |
hormone | ethinylestradiol, progesterone, testosterone |
gastrointestinal agents | cisapride |
histamine H1 antagonists | astemizole, fexofenadine, terfenadine |
immunosuppressives | cyclosporine, sirolimus, tacrolimus |
opoid analgesics | alfentanil, fentanyl, sufentanil |
xanthine | theophylline |
erectile dysfunction drugs | sildenafil, tadalafil |
From “The Grapefruit Challenge,”AJN, Dec. 2004 & The Handbook of Drug-Nutrient Interaction, 2004